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Found 4 of ic50 data for polymerid = 50007499
TargetVoltage-dependent L-type calcium channel subunit beta-2(Homo sapiens)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50101971(BAY-E-9736 | CHEBI:7575 | Nimodipine | Nimotop)
Affinity DataIC50:  30nMAssay Description:Inhibition of human alpha1c/beta2a/alpha2delta1 Cav1.2 expressed in HEK293 cells assessed as Ca2+ current at -80 mV holding potential by patch clamp ...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetVoltage-dependent L-type calcium channel subunit beta-2(Homo sapiens)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50602415(CHEMBL5190568)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of human alpha1c/beta2a/alpha2delta1 Cav1.2 expressed in HEK293 cells assessed as effect on calcium flux by FLIPR analysisMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetVoltage-dependent L-type calcium channel subunit beta-2(Homo sapiens)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50573712(CHEBI:66722 | CHEMBL71260)
Affinity DataIC50:  4.13E+4nMAssay Description:Inhibition of human alpha1c/beta2a/alpha2delta1 Cav1.2 expressed in HEK293 cells assessed as time course of inhibition of membrane potential measured...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit beta-2(Homo sapiens)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50573711(CHEMBL4874732)
Affinity DataIC50:  6.73E+4nMAssay Description:Inhibition of human alpha1c/beta2a/alpha2delta1 Cav1.2 expressed in HEK293 cells assessed as time course of inhibition of membrane potential measured...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed